Glycosidase Inhibitors

Research output

Research output per year 1990 1999 2003 2006

• 28 Article
• 14 (Old data) Lecture or Presentation
• 3 Book
• 3 Chapter

Research output per year

Research output per year

Search results

• 2006

  Fluorescent glycosidase inhibiting 1,5-dideoxy-1,5-iminoalditols

  Greimel, P., Häusler, H., Lundt, I., Rupitz, K., Stütz, A., Tarling, C., Withers, S. G. & Wrodnigg, T. M., 2006, In: Bioorganic & Medicinal Chemistry Letters. 16, 8, p. 2067-2070

  Research output: Contribution to journal › Article › peer-review

• Fluorescently tagged iminoalditol glycosidase inhibitors as novel biological probes and diagnostics

  Lundt, I., Steiner, A., Stütz, A., Tarling, C. A., Ully, S., Withers, S. G. & Wrodnigg, T. M., 2006, In: Bioorganic & Medicinal Chemistry. 14, p. 1737-1742

  Research output: Contribution to journal › Article › peer-review

• L-Idoseptanosides: substrates of D-glucosidases

  Tauss, A., Rupitz, K., Steiner, A., Stütz, A., Tarling, C. A., Withers, S. G. & Wrodnigg, T. M., 2006, In: Tetrahedron / Asymmetry. 17, p. 234-239

  Research output: Contribution to journal › Article › peer-review

• 2005

  Non-natural aldofuranosides as substrates of a beta-glucosidase

  Tauss, A., Greimel, P., Rupitz, K., Steiner, A., Stütz, A., Withers, S. G. & Wrodnigg, T. M., 2005, In: Tetrahedron / Asymmetry. 16, p. 159-165

  Research output: Contribution to journal › Article › peer-review

• 2004

  Golgi endomannosidase inhibitor, alpha-D-glucopyranosyl-(1-3)-1-deoxynojirimycin: A five step synthesis from maltulose and examples of N-modified derivatives

  Spreitz, J. & Stütz, A., 2004, In: Carbohydrate Research. 339, p. 1823-1827

  Research output: Contribution to journal › Article › peer-review

• Simple syntheses of 4-O-glucosylated 1-deoxynojirimycins from maltose and cellobiose

  Steiner, A. & Stütz, A., 2004, In: Carbohydrate Research. 339, 15, p. 2615-2619

  Research output: Contribution to journal › Article › peer-review

• 2002

  A simple method for the preparation of 1-deoxynojirimycin from D-fructose

  Spreitz, J. & Stütz, A., 2002, In: Carbohydrate Research. 337, p. 183-186

  Research output: Contribution to journal › Article › peer-review

• N-Alkylated Derivatives of 1,5-Dideoxy-1,5-iminoxylitol as beta-Xylosidase and beta-Glucosidase Inhibitors

  Häusler, H., Rupitz, K., Stütz, A. & Withers, S. G., 2002, In: Monatshefte für Chemie - Chemical Monthly. 133, p. 555-560

  Research output: Contribution to journal › Article › peer-review

• 2001

  Novel lipophilic derivatives of 2,5-dideoxy-2,5-imino-D-mannitol (DMDP) are powerful beta-glucosidase inhibitors

  Wrodnigg, T. M., Withers, S. G. & Stütz, A., 2001, In: Bioorganic & Medicinal Chemistry Letters. 11, p. 1063-1064

  Research output: Contribution to journal › Article › peer-review

• Powerful probes for glycosidases: Novel fluorescently tagged glycosidase inhibitors

  Hermetter, A., Scholze, H., Stütz, A., Withers, S. G. & Wrodnigg, T. M., 2001, In: Bioorganic & Medicinal Chemistry Letters. 11, p. 1339-1342

  Research output: Contribution to journal › Article › peer-review

• 2000

  Biologically active 1-aminodeoxy derivatives of the powerful glucosidase inhibitor 2,5-dideoxy-2,5-imino-D-mannitol

  Wrodnigg, T. M., Gaderbauer, W., Greimel, P., Häusler, H., Sprenger, F., Stütz, A., Virgona, C. & Withers, S. G., 2000, In: Journal of Carbohydrate Chemistry. 19, p. 975-990

  Research output: Contribution to journal › Article › peer-review

• Syntheses of sugar related trihydroxyazepanes from simple carbohydrates and their activities as reversible glycosidase inhibitors

  Andersen, S. M., Ekhart, C., Lundt, I. & Stütz, A., 2000, In: Carbohydrate Research. 326, p. 22-33

  Research output: Contribution to journal › Article › peer-review

• 1999

  Chemical and chemo-enzymatic approaches to unnatural ketoses and glycosidase inhibitors with basic nitrogen in the sugar ring

  Fechter, M., Stütz, A. & Tauss, A., 1999, In: Current Organic Chemistry . 3, p. 235-251

  Research output: Contribution to journal › Article › peer-review

• 1998

  Synthesis of regio- and stereospecifically C-deuterated derivatives of glycosidase inhibitors 1-deoxymannojirimycin and 2,5-dideoxy-2,5-imino-D-mannitol by intramolecular reductive amination employing deuterium gas

  Berger, A., Fechter, M., Gradnig, G., Mirtl, C., Schmid, W. & Stütz, A., 1998, In: Carbohydrate Research. 309, p. 367-374

  Research output: Contribution to journal › Article › peer-review

• 1997

  Chemical and chemo-enzymatc approaches to glycosidase inhibitors with basic nitrogen in the sugar ring

  De Raadt, A., Ebner, M., Ekhart, C. & Stütz, A., 1997, In: Topics in Current Chemistry. 187, p. 157-186

  Research output: Contribution to journal › Article › peer-review

• Synthesis of 1-amino-1,2,5-trideoxy-2,5-imino-D-mannitol, a novel analogue of the powerful glucosidase inhibitor 2,5-dideoxy-2,5-imino-D-mannitol, via an Amadori rearrangement of 5-azido-5-deoxy-D-glucofuranose

  Stütz, A., Withers, S. G. & Wrodnigg, T. M., 1997, In: Tetrahedron Letters. 38, p. 5463-5466

  Research output: Contribution to journal › Article › peer-review

• Synthesis of a novel alpha-glucoside of the powerful glucosidase inhibitor 2,5-dideoxy-2,5-imino-D-mannitol via enzymatic glucosylation of 5-azido-5-deoxy-D-glucofuranose

  Dax, K., Ebner, M., Peinsipp, R. & Stütz, A., 1997, In: Tetrahedron Letters. 38, p. 225-226

  Research output: Contribution to journal › Article › peer-review

• Two isosteric fluorinated derivatives of the powerful glucosidase inhibitors 1-deoxynojirimycin and 2,5-dideoxy-2,5-imino-D-mannitol: Syntheses and glucosidase inhibitory activities of 1,2,5-trideoxy-2-fluoro-1,5-imino-D-glucitol and of....

  Andersen, S., Ebner, M., Ekhart, C., Gradnig, G., Legler, G., Lundt, I., Stütz, A., Withers, S. G. & Wrodnigg, T. M., 1997, In: Carbohydrate Research. 301, p. 155-166

  Research output: Contribution to journal › Article › peer-review

• 1996

  A novel approach to the 1-deoxynojirimycin system: Synthesis, from sucrose, of 2-acetamido-1,2-dideoxynojirimycin as well as some 2-N-modified derivatives

  Gradnig, G., Legler, G. & Stütz, A., 1996, In: Carbohydrate Research. 287, p. 49-57

  Research output: Contribution to journal › Article › peer-review

• A novel innovative approach aims to clarify the reaction mechanism of retaining glycoside hydrolases

  Stütz, A., 1996, In: Angewandte Chemie - International Edition . 35, p. 1926-1928

  Research output: Contribution to journal › Article › peer-review

• 1995

  Synthesis of (1-13C)-1-deoxynojirimycin

  Berger, A., Ebner, M. & Stütz, A., 1995, In: Tetrahedron Letters. 36, p. 4989-4990

  Research output: Contribution to journal › Article › peer-review

• 1993

  2,5-dideoxy-2,5-imino-D-mannitol and -D-glucitol. Two step bio-organic syntheses from 5-azido-5-deoxy-D-glucofuranose and -L-idofuranose, respectively, evaluation as glucosidase inhibitors and an application in affinity purification and....

  Legler, G., Korth, A., Berger, A., Ekhart, C., Gradnig, G. & Stütz, A., 1993, In: Carbohydrate Research. 250, p. 67-77

  Research output: Contribution to journal › Article › peer-review

• Synthese von (+)-Castanospermin und 1-epi-Castanospermin aus D-Glucofuranurono-6,3-lacton durch Reformatsky-Reaktion

  Grassberger, V., Berger, A., Dax, K., Fechter, M., Gradnig, G. & Stütz, A., 1993, In: Liebigs Annalen der Chemie (1979 - 1994). p. 379-390

  Research output: Contribution to journal › Article › peer-review

• 1992

  A simple and convergent synthesis of the mannosidase inhibitor 1-deoxymannonojirimycin from sucrose

  De Raadt, A. & Stütz, A., 1992, In: Tetrahedron Letters. 33, p. 189-192

  Research output: Contribution to journal › Article › peer-review

• 1991

  First synthesis of (1R,2R,3S,9S,9aR)-1,2,3,9-tetrahydroxyquinolizidine, a novel isosteric homologue of the glucosidase inhibitor castanospermine

  Gradnig, G., Berger, A., Grassberger, V., Legler, G. & Stütz, A., 1991, In: Tetrahedron Letters. 32, p. 4889-4892

  Research output: Contribution to journal › Article › peer-review

• 1990

  Einfache Synthesen von 1,5-didesoxy-1,5-imino-D-glucit (1-Desoxynojirimycin) und 1,6-Didesoxy-1,6-imino-D-glucit aus D-Glucofuranurono-6,3-lacton

  Dax, K., Gaigg, B., Grassberger, V., Kölblinger, B. & Stütz, A., 1990, In: Journal of Carbohydrate Chemistry. 9, p. 479-499

  Research output: Contribution to journal › Article › peer-review

• Einfache Synthese von 1,5,6-Tridesoxy-6-fluor-1,5-imino-D-glucit, dem ersten fluorhältigen Derivat des Glucosidaseninhibitors 1-Desoxynojirimycin

  Dax, K., Grassberger, V. & Stütz, A., 1990, In: Journal of Carbohydrate Chemistry. 9, p. 903-908

  Research output: Contribution to journal › Article › peer-review

• Hexa-O-benzyl-5-hydroxy-pseudo-alpha-D-glucopyranose and its C-5 epimer

  Ferrier, R. J. & Stütz, A., 1990, In: Carbohydrate Research. 205, p. 283-291

  Research output: Contribution to journal › Article › peer-review